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93

抑制剂 & 化合物

20

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Cat. No. Product Name Target Signaling Pathways
T1005 Amoxicillin

Amoxycillin,阿莫西林

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin (Amoxycillin) 是一种具有广谱抗菌活性和良好口服吸收的抗生素。
T9000 Pyrimorph

Antifungal Microbiology/Virology
Pyrimorph 是一种杀真菌剂,对 oomycetes 具有良好抑菌活性。
T10411 AU1235

Antibacterial Microbiology/Virology
AU1235是金刚烷脲,是一种MmpL3抑制剂。结核分枝杆菌蛋白MmpL3在细胞壁合成中起重要作用,它影响海藻糖单支霉菌酸酯跨内膜转运。
T6385 Amoxicillin Sodium

阿莫西林钠,Clavulanate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin Sodium (Clavulanate) 是一种有广谱抗菌活性,口服吸收好的抗生素。它能抑制细胞壁中多肽的生物合成,可抑制细胞生长。
T1008 Cephalexin

头孢氨苄,Cefalexin,Cephacillin

Antibacterial; Antibiotic Microbiology/Virology
Cephalexin (Cephacillin) 是一种强口服活性的头孢菌素抗生素。它通过破坏细菌细胞壁的生长来杀死革兰氏阳性和一些革兰氏阴性细菌。它可研究肺炎、链球菌性咽喉炎、细菌性心内膜炎等。
T2691 Oritavancin diphosphate

奥利万星二磷酸盐,LY333328 diphosphate

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Oritavancin diphosphate (LY333328 diphosphate) 是一种新型半合成的糖肽抗生素, 可研究革兰氏阳性菌感染。
T1005L Amoxicillin trihydrate

Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate

Antibacterial; Antibiotic Microbiology/Virology
Amoxicillin trihydrate (Moxaline trihydrate) 是一种中谱β内酰胺抗菌素。
T1799 Caspofungin Acetate

醋酸卡泊芬净,L 743873,Cancidas,MK 0991,L 743872

Antibiotic; Antifungal Microbiology/Virology
Caspofungin Acetate (MK 0991) 是一种抗真菌药,能够非竞争性地抑制 1,3-β-D 葡聚糖合酶的合成。
T1213 Piperacillin sodium

哌拉西林钠,Sodium piperacillin,CL227193,Piperacillin sodium salt

Antibacterial; Antibiotic Microbiology/Virology
Piperacillin sodium salt(CL227193) )是一种β-内酰胺类广谱抗生素。
T1122 Cephalothin sodium

头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin

Antibacterial; Antibiotic Microbiology/Virology
Cephalothin sodium (Cefalotin) 是一种头孢类抗生素, 具有广泛的抗菌活性,抑制革兰氏阳性和阴性菌。
T1228 Cefonicid sodium

Monocid sodium,头孢尼西钠,Cefonicid disodium salt

Antibacterial; Antibiotic Microbiology/Virology
Cefonicid sodium (Monocid sodium) 是一种广谱头孢类抗生素, 能抑制细菌细胞壁的形成。
T6437 Cefoperazone

头孢哌酮,Cefob,Medocef

Antibacterial; Antibiotic Microbiology/Virology
Cefoperazone (Medocef) 是一种半合成的头孢菌素,有抗菌活性。
T32237 Isoxaben

EL 107,NA 8318,Isoxaben; EL 107; NA 8318

Cell wall Immunology/Inflammation
Isoxaben (EL 107) 是一种细胞壁生物合成的特异性抑制剂,常作为除草剂使用,可抑制放射性标记的葡萄糖掺入酸不溶性细胞壁部分。
T19595 UDP-glucuronic acid trisodium

尿苷二磷酸葡萄糖醛酸三钠,UDP-​glucuronic acid trisodium,尿苷二磷酸葡糖醛酸

Others Others
UDP-glucuronic acid trisodium (UDP-​glucuronic acid trisodium) is an indispensable precursor for vital glycoconjugates in various biological domains. These glycoconjugates encompass mammalian glycosaminoglycans, plant cell wall polysaccharides, and bacterial capsule glycoglycerolipids.
T1224 Cefuroxime sodium

Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin

Antibacterial; Antibiotic Microbiology/Virology
Cefuroxime sodium (Cefuroxime sodium salt) 是一种具有口服活性的头孢菌素抗生素,增加了对 β-内酰胺酶的稳定性。
T0953 Cefazolin sodium

Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazolin sodium (cephazolin sodium) salt 是一种头孢类抗生素, 可研究多种细菌感染。
T6386 Ampicillin sodium

氨苄西林钠,Domicillin,D-(-)-α-Aminobenzylpenicillin sodium salt,Penialmen,Citteral

Antibacterial; Antibiotic Microbiology/Virology
Ampicillin sodium (Domicillin) 是Ampicillin 的钠盐形式,是Ampicillin 的广谱半合成衍生物。它通过与青霉素结合蛋白结合来抑制细菌细胞壁的合成,从而抑制肽聚糖的合成,肽聚糖是细菌细胞壁的关键成分。
T1063 Ticarcillin disodium

Ticarpen,Ticarcillin disodium salt,替卡西林二钠

Antibacterial; Antibiotic Microbiology/Virology
Ticarcillin disodium (Ticarpen) 主要用于抗革兰氏阴性菌, 特别是绿脓杆菌, 也是少数可研究嗜麦芽感染的抗生素。
T0932 Cefixime

FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635

Antibacterial; Antibiotic Microbiology/Virology
Cefixime (FR-17027) 是一种头孢菌素类抗生素, 可研究一些细菌感染。
T5022 Ceforanide

Antibacterial; Antibiotic Microbiology/Virology
Ceforanide 是一种头孢菌素,可静脉或肌肉给药。它在体外具有一系列抗菌活性。
T1616 Cefotiam hydrochloride

盐酸头孢替安,Pansporin,SCE-963 hydrochloride,Pansporine,头孢替安盐酸盐,Cefotiam dihydrochloride,Halospor

Antibacterial; Antibiotic Microbiology/Virology
Cefotiam hydrochloride (SCE-963 hydrochloride) 是一种肠外头孢菌素类广谱抗生素,对革兰氏阳性菌和革兰氏阴性菌有活性。
T4202 Delamanid

迪拉马尼,德拉马尼,OPC-67683

Anti-infection; Antibacterial; Antibiotic Microbiology/Virology
Delamanid (OPC-67683) 是一种新的分枝杆菌细胞壁合成抑制剂,可用于耐多药结核病。
T14386 AZD9567

Mizacorat

Glucocorticoid Receptor Endocrinology/Hormones
AZD9567 是一种强效且具有口服活性和选择性的非类固醇糖皮质激素受体调节剂(SGRM),其 IC50 值为 3.8 nM。它在链球菌细胞壁(SCW)再活化关节炎症模型中显示出卓越的疗效。
T2213 Terconazole

Gyno-Terazol,Terazol 3,Terazol 7,Triaconazole,特康唑,曲康唑,R42470

Antifection; Antifungal Microbiology/Virology
Terconazole (Terazol 7) 是一种广谱抗真菌药物,用于研究阴道酵母菌感染。
T12470 Picloxydine

Antibacterial Microbiology/Virology
Picloxydine 是一种杂环双胍,有抗细菌和牙菌斑活性。
T3131 Fosfomycin calcium

Phosphomycin calcium salt,Fosmicin,磷霉素钙

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin calcium (Phosphomycin calcium salt) 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药细菌。
T1451 Levofloxacin hydrate

左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Levofloxacin hydrate (Cravit hydrate) 是抗生素化合物,抑制细菌DNA 旋转酶活性。
T7043 Cefotetan

头孢替坦,Apacef

Antibacterial; Antibiotic Microbiology/Virology
Cefotetan (Apacef) 是一种半合成的头霉素抗生素,能抑制细胞壁合成发挥杀菌作用。
T61355 APX2039

APX-2039,APX 2039

Antifungal Microbiology/Virology
APX2039 是一种口服有效的真菌 Gwt1 酶 (fungal Gwt1 enzyme) 抑制剂,是新型Gwt2096抑制剂APX1的前药。APX2039 对 C. neoformans 和 C. gattii 展现出极强的抗氪球菌活性。APX2039 具有有效的抗真菌活性,科阻断 GPI (糖基磷脂酰肌醇)锚定细胞壁甘露蛋白的定位。APX2039 可用于研究隐球菌脑膜炎 (CM) 。
T19721 Epoxiconazole

BAS-480F,BAS 480F,EC 406 850 2,氟环唑,BAS480F,EC-406-850-2

Antifungal Microbiology/Virology
Epoxiconazole (BAS-480F) 是一种 14-α 去甲基化酶抑制剂,抑制麦角甾醇的合成和真菌细胞壁的形成。它是一种杀菌剂,对耐多菌灵和耐苯甲酰胺的菌株均表现出强大的抑制作用,可用于控制多种农作物病害。
T61194 D75-4590

Others Others
D75-4590是一种β-1,6-葡聚糖抑制剂。由于葡聚糖是细胞壁的主要成分,特别是β-1,6-葡聚糖,D75-4590可以通过抑制其合成酶来对抗真菌感染。
T7858 Ceftezole sodium

Celoslin,Falomesin,头孢替唑钠,Alomen

Anti-infection; Antibacterial; Antibiotic; Glucosidase Metabolism; Microbiology/Virology
Ceftezole sodium (Falomesin) 是一种广谱 cephem 抗生素,具有抑制多种革兰氏阳性菌和革兰氏阴性菌活性。它是一种α-葡萄糖苷酶抑制剂,具有体内抗糖尿病活性。
T6686 Sulconazole mononitrate

Exelderm,Sulconazole Nitrate,RS 44872,硝酸硫康唑

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Sulconazole mononitrate (Exelderm) 是一种咪唑类广谱杀菌剂。它可研究皮肤真菌病,花斑糠疹病,皮肤念珠菌病。
T1482 Ciclopirox

环吡酮,HOE296b,环吡酮胺

ATPase; Ferroptosis; Antibacterial; Autophagy; Antifungal Apoptosis; Autophagy; Membrane transporter/Ion channel; Microbiology/Virology
Ciclopirox (HOE296b) 是一种合成的抗真菌剂,可研究浅表真菌病。
T8747 Levofloxacin hydrochloride

DNA gyrase; Topoisomerase DNA Damage/DNA Repair
Levofloxacin hydrochloride 是一种广谱的第三代氟喹诺酮类抗生素,是氧氟沙星的光学活性 L-异构体,具有抗菌活性。左氧氟沙星通过细菌细胞壁扩散并通过抑制 DNA 促旋酶(细菌拓扑异构酶 II)起作用,这是一种 DNA 复制、RNA 转录和细菌 DNA 修复所需的酶。 DNA 促旋酶活性的抑制导致细菌细胞生长受阻。
T5024 Cefotiam Hexetil Hydrochloride

盐酸头孢替安酯,头孢替安海替酯盐酸盐

Antibacterial; Antibiotic Microbiology/Virology
Cefotiam hexetil hydrochloride 是一种可口服头孢菌素,是抗生素 cefotiam 的前药,但无抗菌作用。
T11888 LtaS-IN-1

Others; Antibacterial Microbiology/Virology; Others
LtaS-IN-1 是多药耐药粪肠球菌中脂磷壁酸合成的有效抑制剂,可改变细胞壁形态。 LtaS-IN-1 对抗肠球菌属 28 菌株,MIC 值从 0.5 μg/mL 到 64 μg/mL 不等。 LtaS-IN-1 抑制菌株 E1630 和 E1590,MIC 值为 0.5 μg/mL。
T1600 Doxifluridine

Ro 21-9738,AMC 0101,5'-DFUR,5-Fluoro-5'-deoxyuridine,去氧氟尿苷

Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Doxifluridine (AMC 0101) 是一种胸苷磷酸化酶活化剂,对 PC9-DPE2细胞的 IC50为0.62 μM。它是具有抗肿瘤活性的抗肿瘤剂 5-fluorouracil (5-FU) 的氟嘧啶衍生物和口服前药。
T32206 Isodityrosine

Isodityrosine is a new cross-linking amino acid from plant cell-wall glycoprotein.
T27813 Lenapenem

carbapenem

Lenapenem is a broad-spectrum, carbapenem antibiotic with bactericidal activity by weakens the bacterial cell wall and leads to lytic cell death.
T69266 Cefcanel free acid

Cefcanel is a semisynthetic third-generation cephalosporin with antibacterial activity. Cefcanel is active against the species E. coli, K. aerogenes and Proteus mirabilis; H. influenzae and M. catarrhalis has reasonable susceptibility. Cefcanel inhibits 90% of S. aureus strains at 2 µg/ml, irrespective of the presence of a β-lactamase. Cefcanel binds to and inactivates penicillin-binding proteins (PBPs) located on the inner membrane of the bacterial cell wall. PBPs are enzymes involved in the te...
T25221 Cefaparole

Cefaparol,Lilly 110264,Lilly-110264,Lilly110264,Cefaparolum

Cefaparole is an antibacterial compound and cell wall biosynthesis inhibitor.
T69454 Cephradine dihydrate

Cephradine dihydrate is the hydrate form of Cephradine (free base), a semi-synthetic cephalosporin antibiotic. Cefradin inhibits the last stage of bacterial cell wall synthesis by binding to certain penicillin-binding proteins which results in cell lysis. Cell lysis is mediated by bacterial cell wall autolytic enzymes. Cefradin may interfere with autolysin inhibitors.
T68780 Puupehenone

Puupehenone is a natural heat shock protein 90 (Hsp90) inhibitor, potentiating the echinocandin drug caspofungin in caspofungin-resistant fungal pathogens, blocking the induction of caspofungin-responding genes required for the adaptation to cell wall stress through the cell wall integrity (CWI) pathway.
T20897 Cefepime dihydrochloride

Cefepime hydrochloride anhydrous,BMY-28142 dihydrochloride,Cepimax,Axepim,Cefepime HCl

Cefepime dihydrochloride, a broad-spectrum fourth-generation cephalosporin, binds and inactivates penicillin-binding proteins (PBPs) located on the inner membrane of the bacterial cell wall.
T25267 Cmpd 339509

Cmpd339509,Cmpd-339509

Cmpd 339509 is a DprE1 inhibitor. DprE1 is an epimerase required for cell wall biosynthesis.
T27390 Friulimicin B

Friulimicin B is a peptidoglycan synthesis inhibitor with excellent activity against gram-positive pathogens through cell wall interruption.
T4995L Cefpirome

Cefpiromum,HR 810,HR810,Cefpiroma,HR-810

Cefpirome is a broad-spectrum, fourth-generation cephalosporin. It binds to and inactivates penicillin-binding proteins located on the inner membrane of the bacterial cell wall.
T71341 Myclobutanil hydroxide

Myclobutanil hydroxide is a 14-α demethylase inhibitor that inhibits ergosterol synthesis and fungal cell wall formation. It also weakly inhibits testosterone production.
T68777 FR-900148 sodium dihydrate

FR-900148 sodium dihydrate is an antibiotic that inhibits cell wall synthesis.

化合物

Amoxicillin
Cat.No: T1005
Synonym: Amoxycillin,阿莫西林
Target: Antibacterial, Antibiotic
Pyrimorph
Cat.No: T9000
Synonym:
Target: Antifungal
AU1235
Cat.No: T10411
Synonym:
Target: Antibacterial
Amoxicillin Sodium
Cat.No: T6385
Synonym: 阿莫西林钠,Clavulanate
Target: Antibacterial, Antibiotic
Cephalexin
Cat.No: T1008
Synonym: 头孢氨苄,Cefalexin,Cephacillin
Target: Antibacterial, Antibiotic
Oritavancin diphosphate
Cat.No: T2691
Synonym: 奥利万星二磷酸盐,LY333328 diphosphate
Target: Others, Antibacterial, Antibiotic
Amoxicillin trihydrate
Cat.No: T1005L
Synonym: Amoxycillin trihydrate,Amoxil trihydrate,Amoxipen trihydrate,阿莫西林三水物,Moxaline trihydrate
Target: Antibacterial, Antibiotic
Caspofungin Acetate
Cat.No: T1799
Synonym: 醋酸卡泊芬净,L 743873,Cancidas,MK 0991,L 743872
Target: Antibiotic, Antifungal
Piperacillin sodium
Cat.No: T1213
Synonym: 哌拉西林钠,Sodium piperacillin,CL227193,Piperacillin sodium salt
Target: Antibacterial, Antibiotic
Cephalothin sodium
Cat.No: T1122
Synonym: 头孢噻吩钠,Cefalotin sodium,Cephalothin,Cefalotin
Target: Antibacterial, Antibiotic
Cefonicid sodium
Cat.No: T1228
Synonym: Monocid sodium,头孢尼西钠,Cefonicid disodium salt
Target: Antibacterial, Antibiotic
Cefoperazone
Cat.No: T6437
Synonym: 头孢哌酮,Cefob,Medocef
Target: Antibacterial, Antibiotic
Isoxaben
Cat.No: T32237
Synonym: EL 107,NA 8318,Isoxaben; EL 107; NA 8318
Target: Cell wall
UDP-glucuronic acid trisodium
Cat.No: T19595
Synonym: 尿苷二磷酸葡萄糖醛酸三钠,UDP-​glucuronic acid trisodium,尿苷二磷酸葡糖醛酸
Target: Others
Cefuroxime sodium
Cat.No: T1224
Synonym: Anaptivan,头孢呋辛钠,Cefuroxime sodium salt,Biociclin
Target: Antibacterial, Antibiotic
Cefazolin sodium
Cat.No: T0953
Synonym: Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin
Target: Others, Antibacterial, Antibiotic
Ampicillin sodium
Cat.No: T6386
Synonym: 氨苄西林钠,Domicillin,D-(-)-α-Aminobenzylpenicillin sodium salt,Penialmen,Citteral
Target: Antibacterial, Antibiotic
Ticarcillin disodium
Cat.No: T1063
Synonym: Ticarpen,Ticarcillin disodium salt,替卡西林二钠
Target: Antibacterial, Antibiotic
Cefixime
Cat.No: T0932
Synonym: FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635
Target: Antibacterial, Antibiotic
Ceforanide
Cat.No: T5022
Synonym:
Target: Antibacterial, Antibiotic
Cefotiam hydrochloride
Cat.No: T1616
Synonym: 盐酸头孢替安,Pansporin,SCE-963 hydrochloride,Pansporine,头孢替安盐酸盐,Cefotiam dihydrochloride,Halospor
Target: Antibacterial, Antibiotic
Delamanid
Cat.No: T4202
Synonym: 迪拉马尼,德拉马尼,OPC-67683
Target: Anti-infection, Antibacterial, Antibiotic
AZD9567
Cat.No: T14386
Synonym: Mizacorat
Target: Glucocorticoid Receptor
Terconazole
Cat.No: T2213
Synonym: Gyno-Terazol,Terazol 3,Terazol 7,Triaconazole,特康唑,曲康唑,R42470
Target: Antifection, Antifungal
Picloxydine
Cat.No: T12470
Synonym:
Target: Antibacterial
Fosfomycin calcium
Cat.No: T3131
Synonym: Phosphomycin calcium salt,Fosmicin,磷霉素钙
Target: Antibacterial, Antibiotic
Levofloxacin hydrate
Cat.No: T1451
Synonym: 左氧氟沙星半水合物,Levaquin hydrate,Cravit hydrate,Quixin hydrate,Levofloxacin Hemihydrate,Tavanic hydrate,Iquix hydrate
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Cefotetan
Cat.No: T7043
Synonym: 头孢替坦,Apacef
Target: Antibacterial, Antibiotic
APX2039
Cat.No: T61355
Synonym: APX-2039,APX 2039
Target: Antifungal
Epoxiconazole
Cat.No: T19721
Synonym: BAS-480F,BAS 480F,EC 406 850 2,氟环唑,BAS480F,EC-406-850-2
Target: Antifungal
D75-4590
Cat.No: T61194
Synonym:
Target: Others
Ceftezole sodium
Cat.No: T7858
Synonym: Celoslin,Falomesin,头孢替唑钠,Alomen
Target: Anti-infection, Antibacterial, Antibiotic, Glucosidase
Sulconazole mononitrate
Cat.No: T6686
Synonym: Exelderm,Sulconazole Nitrate,RS 44872,硝酸硫康唑
Target: Antibacterial, Antibiotic, Antifungal
Ciclopirox
Cat.No: T1482
Synonym: 环吡酮,HOE296b,环吡酮胺
Target: ATPase, Ferroptosis, Antibacterial, Autophagy, Antifungal
Levofloxacin hydrochloride
Cat.No: T8747
Synonym:
Target: DNA gyrase, Topoisomerase
Cefotiam Hexetil Hydrochloride
Cat.No: T5024
Synonym: 盐酸头孢替安酯,头孢替安海替酯盐酸盐
Target: Antibacterial, Antibiotic
LtaS-IN-1
Cat.No: T11888
Synonym:
Target: Others, Antibacterial
Doxifluridine
Cat.No: T1600
Synonym: Ro 21-9738,AMC 0101,5'-DFUR,5-Fluoro-5'-deoxyuridine,去氧氟尿苷
Target: Nucleoside Antimetabolite/Analog, DNA/RNA Synthesis
Isodityrosine
Cat.No: T32206
Synonym:
Target:
Lenapenem
Cat.No: T27813
Synonym: carbapenem
Target:
Cefcanel free acid
Cat.No: T69266
Synonym:
Target:
Cefaparole
Cat.No: T25221
Synonym: Cefaparol,Lilly 110264,Lilly-110264,Lilly110264,Cefaparolum
Target:
Cephradine dihydrate
Cat.No: T69454
Synonym:
Target:
Puupehenone
Cat.No: T68780
Synonym:
Target:
Cefepime dihydrochloride
Cat.No: T20897
Synonym: Cefepime hydrochloride anhydrous,BMY-28142 dihydrochloride,Cepimax,Axepim,Cefepime HCl
Target:
Cmpd 339509
Cat.No: T25267
Synonym: Cmpd339509,Cmpd-339509
Target:
Friulimicin B
Cat.No: T27390
Synonym:
Target:
Cefpirome
Cat.No: T4995L
Synonym: Cefpiromum,HR 810,HR810,Cefpiroma,HR-810
Target:
Myclobutanil hydroxide
Cat.No: T71341
Synonym:
Target:
FR-900148 sodium dihydrate
Cat.No: T68777
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
PDK0101 4-Methylcinnamic acid

对甲基肉桂酸,对甲基肉桂

Antifungal Microbiology/Virology
4-Methylcinnamic acid 是一种肉桂酸类似物,可用作克服抗真菌耐受性的干预催化剂。它可提高细胞壁破坏剂的效力。
T1165 Ethionamide

Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide

Dehydrogenase; CAT; Antibacterial; Antibiotic Metabolism; Microbiology/Virology; oxidation-reduction
Ethionamide (2-ethylthioisonicotinamide) 是一种抗结核抗生素。
T0810 Ethambutol dihydrochloride

Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Ethambutol dihydrochloride (CL40881) 能抗分枝杆菌,可抑制阿拉伯糖基转移酶活性来阻止细胞壁形成。
T1226 Bacitracin

Albac,Ziba-RX,杆菌肽

Antibacterial; Antibiotic Microbiology/Virology
Bacitracin (Ziba-RX) 是一种用于葡萄球菌感染的多肽抗生素。它通过与焦磷酸十一癸烯基结合,起抑制细胞壁生物合成作用。
T0146 Tioconazole

UK-20349,Vagistat,噻康唑

Antibiotic; Antifection; Antifungal Microbiology/Virology
Tioconazole (Vagistat) 是一种广谱性的抗真菌咪唑衍生物。它抑制几种皮肤真菌和几种酵母菌的 MIC50分别小于 3.12 mg/L 和 9 mg/L。
T40646 Lipoteichoic acid

Complement System Immunology/Inflammation
Lipoteichoic acid 是 Staphylococcus aureus 细胞壁的聚合物,通过诱导 C3 和抑制 CD55 来激活补体系统,通过 IGF-1 途径减少脂肪沉积。
T6S0920 2"-O-Galloylhyperin

2”-O-没食子酰基金丝桃苷,2''-O-Galloylhyperin,Q-100605,FT-0689359

Others Others
2"-O-Galloylhyperin (FT-0689359) 是一种分离自Pyrola incarnateFisch. 中的活性化合物,具有抗氧化和抗炎作用,对氧化应激诱导的肝损伤具有肝保护作用。
T8262 Fosfomycin sodium

Fosfomycin Disodium,磷霉素钠

Antibacterial; Antibiotic Microbiology/Virology
Fosfomycin sodium 是一种能透过血脑屏障的广谱抗生素,不可逆地抑制细胞壁合成的早期阶段。它对多种细菌具有杀菌活性,包括耐多药、广泛耐药和耐全药的细菌。
T1313 Nitrofurantoin

Furadantine,呋喃妥因,Macrodantin,Furadonine

Antibacterial; Antibiotic Microbiology/Virology
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。
TN1569 Deoxylapachol

Antifection; Antifungal Microbiology/Virology
Deoxylapachol 是新西兰褐藻Landsburgia quercifolia 的主要细胞毒性成分,有抗真菌和抗癌活性。
T4889 2,6-Diaminoheptanedioic acid

Others; Endogenous Metabolite Metabolism; Others
2,6-Diaminoheptanedioic acid 是内源性代谢产物的一种。
T27237 Echinocandin B

A-30912A,NSC 287461,A 30912A,A30912A,A22082

Echinocandin B is a cyclic hexapeptide echinocandin antibiotic from Aspergillus nidulans var. echinulatus . It attacks the cell wall of fungi by inhibiting beta-1,3-glucan synthesis.
T40814 Colominic acid sodium salt

Polysialic acid sodium salt,Colominic acid sodium salt

Colominic acid sodium salt, also known as polysialic acid sodium salt, is naturally isolated from the cell wall of Escherichia coli and animals. It exhibits a red color with an absorption maximum of 530 nm and possesses anti-bacterial activity.
T4984 Cefozopran hydrochloride

SCE-2787 hydrochloride

Antifungal Microbiology/Virology
Cefozopran hydrochloride (SCE-2787 hydrochloride) 是一种半合成的非肠道头孢菌素。它是一种广谱抗菌抗生素,能抑制大多数革兰氏阴性和革兰氏阳性菌。
T75686 Enfumafungin

Enfumafungin,一种从Hormonema carpetanum菌提取的三萜糖苷,具有抗真菌特性,主要通过作为(1,3)-beta-D-葡聚糖合酶抑制剂影响真菌细胞壁发挥作用。其对酵母和多数真菌(除隐球菌外)有效,但不会抑制枯草芽孢杆菌的生长。
T77242 Pectin

Pectin是从高等植物细胞壁中提取的一种杂多糖。作为纳米颗粒制备,它用作活性分子的运载载体。此外,Pectin还具有吸附剂和广谱抗菌剂的功能,能够结合肠道粘膜中的细菌毒素及其他刺激物,从而缓解受刺激的黏膜。
T78490 Polygalacturonic acid

Galacturonic acid polymer

Polygalacturonic acid(Galacturonic acid polymer)为透明胶状物,构成细胞壁关键组分。该酸应用于制备银纳米颗粒(AgNPs),充当抗氧化剂与抗炎剂,防护细胞遭受ROS增高引起的损伤,并促进伤口愈合。Polygalacturonic acid纳米颗粒亦显示抗菌性能。
T81428 Polypectate sodium

pectate sodium

Polypectate sodium作为细胞壁多糖(果胶)的关键组分,充当碳源及多聚半乳糖醛酸酶诱导剂。此外,Polypectate sodium适用于评估链霉菌属果胶酸裂解酶的碱性活性与稳定性,同时用于黄腐藻多聚半乳糖醛酸酶生产及反应条件的优化研究。
T35751 Violacein

Violacein is a bacterial metabolite originally isolated from C. violaceum that has antibacterial and antiprotozoal activities.[1] [2] It is produced by C. violaceum as a purple pigment in response to N-hexanoyl homoserine lactone , a property that has been modified to create a strain of C. violaceum used in detecting quorum-sensing molecules.[3] Violacein is active against Gram-positive bacteria, including B. subtilis and S. aureus (MICs = 0.8 and 1.6 &#181M, respectively). It is also active aga...
T35624 Ajoene

Ajoene is a disulfide that has been found inA. sativumand has diverse biological activities, including antibacterial, anticancer, antiplatelet, and antioxidant properties.1,2,3,4It is active against Gram-positive (MICs = 5-160 &#181g/ml) and Gram-negative bacteria (MICs = 136-200 &#181g/ml), as well as yeasts (MICs = 10-20 &#181g/ml).1Ajoene is cytotoxic to mouse melanoma cells (IC50= 18 &#181M), as well as human colon, lung, mammary, and pancreatic cancer cells (IC50s = 7-41 &#181M).2It reduces...

天然产物

4-Methylcinnamic acid
Cat.No: PDK0101
Synonym: 对甲基肉桂酸,对甲基肉桂
Target: Antifungal
Ethionamide
Cat.No: T1165
Synonym: Bayer 5312,乙硫异烟胺,2-ethylthioisonicotinamide,Ethinamide
Target: Dehydrogenase, CAT, Antibacterial, Antibiotic
Ethambutol dihydrochloride
Cat.No: T0810
Synonym: Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881
Target: Antibacterial, Antibiotic, Antifungal
Bacitracin
Cat.No: T1226
Synonym: Albac,Ziba-RX,杆菌肽
Target: Antibacterial, Antibiotic
Tioconazole
Cat.No: T0146
Synonym: UK-20349,Vagistat,噻康唑
Target: Antibiotic, Antifection, Antifungal
Lipoteichoic acid
Cat.No: T40646
Synonym:
Target: Complement System
2"-O-Galloylhyperin
Cat.No: T6S0920
Synonym: 2”-O-没食子酰基金丝桃苷,2''-O-Galloylhyperin,Q-100605,FT-0689359
Target: Others
Fosfomycin sodium
Cat.No: T8262
Synonym: Fosfomycin Disodium,磷霉素钠
Target: Antibacterial, Antibiotic
Nitrofurantoin
Cat.No: T1313
Synonym: Furadantine,呋喃妥因,Macrodantin,Furadonine
Target: Antibacterial, Antibiotic
Deoxylapachol
Cat.No: TN1569
Synonym:
Target: Antifection, Antifungal
2,6-Diaminoheptanedioic acid
Cat.No: T4889
Synonym:
Target: Others, Endogenous Metabolite
Echinocandin B
Cat.No: T27237
Synonym: A-30912A,NSC 287461,A 30912A,A30912A,A22082
Target:
Colominic acid sodium salt
Cat.No: T40814
Synonym: Polysialic acid sodium salt,Colominic acid sodium salt
Target:
Cefozopran hydrochloride
Cat.No: T4984
Synonym: SCE-2787 hydrochloride
Target: Antifungal
Enfumafungin
Cat.No: T75686
Synonym:
Target:
Pectin
Cat.No: T77242
Synonym:
Target:
Polygalacturonic acid
Cat.No: T78490
Synonym: Galacturonic acid polymer
Target:
Polypectate sodium
Cat.No: T81428
Synonym: pectate sodium
Target:
Violacein
Cat.No: T35751
Synonym:
Target:
Ajoene
Cat.No: T35624
Synonym:
Target:
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